Neurotransmitter Transporters

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  • DL-TBOA

    DL-TBOA is a competitive, non-transportable blocker of excitatory amino acid transporters (IC50 values are 70, 6, and 6 μM for EAAT1, EAAT2 and EAAT3 respectively), which also inhibits EAAT4 and EAAT5 (Ki values are 4.4 and 3.2 μM respectively). Learn More

    Starting at: $140.00

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  • (±)-HIP-A

    (±)-HIP-A is a potent, non-competitive excitatory amino acid transporter (EAAT) blocker which preferentially inhibits glutamate-induced [3H]D-aspartate release (IC50 = 1.6 μM) rather than [3H]L-glutamate uptake (IC50 = 18 μM). Learn More

    Starting at: $139.00

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  • LY 2365109 hydrochloride

    LY 2365109 hydrochloride is a potent and selective glycine transporter 1 (GlyT1) inhibitor that induces a dose-dependent elevation in CSF levels of glycine, and enhances acetylcholine and dopamine release in the striatum and prefrontal cortex respectively. Learn More

    Starting at: $149.00

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  • Org 24598 lithium salt

    Org 24598 lithium salt is a selective inhibitor of the glial glycine transporter (GlyT1). pIC50 values are 6.9, <4 and <3 for GlyT1, GABA transporter and Glyt2 respectively. Learn More

    Starting at: $139.00

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  • Org 25543 hydrochloride

    Org 25543 hydrochloride is a potent and selective glycine transporter type 2 (GlyT2) inhibitor (IC50 = 16 nM for hGlyT2), which displays no activity at GlyT1 or 56 other common biological targets (≥ 100 μM), in a glycine uptake assay in CHO cells. Learn More

    Starting at: $139.00

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  • NFPS

    NFPS is a selective, non-transportable inhibitor of GlyT1 which displays no activity on GlyT2 or the transport of proline, GABA or glutamate (IC50 values are 2.8, 9.8 and 56000 nM for hGlyT1, rGlyT1 and rGlyT2 respectively). Learn More

    Starting at: $139.00

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  • Sarcosine

    Sarcosine is an endogenous inhibitor of GlyT1 that displays antipsychotic activity. Learn More

    Starting at: $55.00

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  • Dilazep dihydrochloride

    Dilazep dihydrochloride is a coronary and cerebral vasodilator, suppresses the effects of ischemia. Learn More

    Starting at: $90.00

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  • Decynium 22

    Decynium 22 is an inhibitor of the plasma membrane monoamine transporter (PMAT) (Ki = 0.10 μM). Learn More

    Starting at: $49.00

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