Neurotransmitter Transporters

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  • 3α-Bis-(4-fluorophenyl) methoxytropane hydrochloride

    3α-Bis-(4-fluorophenyl) methoxytropane hydrochloride is a potent inhibitor of dopamine uptake and transport (Ki = 11.8 nM). Learn More

    Starting at: $75.00

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  • JHW 007 hydrochloride

    JHW 007 hydrochloride is a dopamine uptake inhibitor which displays high affinity for the dopamine transporter (DAT) (Ki = 25 nM compared to 1330 and 1730 for NET and SERT respectively), and suppresses the effects of cocaine administration in a dose-dependent manner. Learn More

    Starting at: $120.00

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  • 3-CPMT

    3-CPMT binds with high affinity to the dopamine transporter (Ki = 30 nM) and blocks re-uptake of dopamine. Learn More

    Starting at: $50.00

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  • Mephedrone hydrochloride

    Mephedrone hydrochloride Inhibits striatal dopamine uptake and hippocampal 5-HT uptake in synaptosomes (IC50 values are 467 and 558 nM respectively). Learn More

    Starting at: $95.00

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  • BTCP maleate

    BTCP maleate is a potent dopamine re-uptake inhibitor with a behavioral profile different from that of PCP and similar to that of cocaine. Learn More

    Starting at: $95.00

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  • MPDC

    MM 77 dihydrochloride is a highly potent and fairly selective 5-HT1A ligand, which may be a full antagonist at postsynaptic receptors. Learn More

    Starting at: $135.00

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  • Dihydrokainic acid

    Dihydrokainic acid is a EAAT2(GLT1)-selective non-transportable inhibitor of L-glutamate and L-aspartate uptake. Learn More

    Starting at: $49.00

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  • (±)-threo-3-Methylglutamic acid

    (±)-threo-3-Methylglutamic acid is a potent blocker of glutamate transport. Learn More

    Starting at: $89.00

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  • L-trans-2,4-PDC

    L-trans-2,4-PDC is a potent, competitive, transportable EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor. Learn More

    Starting at: $115.00

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  • L-(-)-threo-3-Hydroxyaspartic acid

    L-(-)-threo-3-Hydroxyaspartic acid is a potent, competitive, transportable EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor. Learn More

    Starting at: $149.00

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  • cis-ACBD

    cis-ACBD is a potent, competitive and selective inhibitor of glutamate uptake. Learn More

    Starting at: $99.00

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  • WAY 213613

    WAY 213613 is a potent, non-substrate inhibitor of EAAT2 (GLT-1) that displays > 44-fold selectivity over EAAT1 and EAAT3. Learn More

    Starting at: $139.00

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  • TFB-TBOA

    TFB-TBOA is a high affinity, selective blocker of glial glutamate transporters EAAT1 and EAAT2 (IC50 values are 17, 22 and 300 nM for EAAT2, EAAT1 and EAAT3 respectively), which displays no activity on a wide range of neurotransmitter receptors and transporters. Learn More

    Starting at: $89.00

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  • Evans Blue tetrasodium salt

    Evans Blue tetrasodium salt is a potent inhibitor of L-glutamate uptake into synaptic vesicles, which inhibits AMPA and kainate receptor-mediated currents (IC50 values are 220 and 150 nM respectively). Learn More

    Starting at: $65.00

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  • (±)-HIP-B

    (±)-HIP-B is a potent, non-competitive excitatory amino acid transporter (EAAT) blocker which preferentially inhibits glutamate-induced [3H]D-aspartate release (IC50 = 1.2 μM) rather than [3H]L-glutamate uptake (IC50 = 16.9 μM). Learn More

    Starting at: $139.00

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  • Chicago Sky Blue 6B

    Chicago Sky Blue 6B is a potent inhibitor of L-glutamate uptake into synaptic vesicles, which inhibits macrophage migration inhibitory factor (MIF) (IC50 = 0.81 μM) and MIF proinflammatory activity. Learn More

    Starting at: $49.00

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  • Ceftriaxone disodium salt

    Ceftriaxone disodium salt is β-lactam antibiotic, which increased activity of the EAAT2 glutamate transporter and displays neuroprotective activity in vivo via upregulation. Learn More

    Starting at: $49.00

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  • L-CCG-lll

    L-CCG-lll is a potent and competitive inhibitor of both glial and neuronal uptake of glutamate, aspartate and cysteate. Learn More

    Starting at: $265.00

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  • 7-Chlorokynurenic acid sodium salt

    7-Chlorokynurenic acid sodium salt is a sodium salt of 7-Chlorokynurenic acid, an NMDA receptor antagonist acting at the glycine site. Learn More

    Starting at: $65.00

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  • 7-Chlorokynurenic acid

    7-Chlorokynurenic acid is a NMDA receptor antagonist acting at the glycine site. Potent competitive inhibitor of L-glutamate transport into synaptic vesicles. Learn More

    Starting at: $60.00

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