Ligand-gated Ion Channels
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L-Aspartic acid
L-Aspartic acid is an endogenous NMDA receptor agonist. Learn MoreStarting at: $32.00
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D-AP5
D-AP5 is a competitive NMDA antagonist. Learn MoreStarting at: $59.00
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D-AP7
D-AP7 is a more active form of AP7. Learn MoreStarting at: $179.00
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MNI-caged-D-aspartate
MNI-caged-D-aspartate is a D-aspartate caged with the photosensitive 4-methoxy-7-nitroindolinyl group. Learn MoreStarting at: $149.00
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A 844606
A 844606 is a selective α7 nicotinic acetylcholine receptor (nAChR) agonist with EC50 values of 1.4 and 2.2 μM at human and rat receptors respectively. Learn MoreStarting at: $129.00
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SEN 12333
SEN 12333 is a α7 nicotinic acetylcholine receptor (nAChR) agonist that displays functional antagonism at histamine H3 receptors (IC50 = 103 nM) and weak agonist activity at human ganglionic α3 nAChRs with an IC50 value of 8.5 μM. Learn MoreStarting at: $125.00
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Quinolinic acid
Quinolinic acid is an endogenous NMDA agonist and transmitter candidate. Learn MoreStarting at: $59.00
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LY 2087101
LY 2087101 is an allosteric potentiator of α7, α4β2 and α4β4 nAChRs. Learn MoreStarting at: $125.00
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CCMI
CCMI is a positive allosteric modulator of α7 neuronal nicotinic acetylcholine receptors (nAChR) that evokes positive modulation of acetylcholine (ACh)-induced EC5 currents. Learn MoreStarting at: $95.00
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L-AP5
L-AP5 is a NMDA antagonist and also an agonist at quisqualate-sensitized AP6 site. Learn MoreStarting at: $145.00
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DL-AP7
DL-AP7 is a phosphono NMDA antagonist. Learn MoreStarting at: $79.00
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Dextromethorphan hydrobromide
Dextromethorphan hydrobromide is a Non-competitive, low affinity NMDA receptor antagonist with the effect of antitussive, anticonvulsive and neuroprotective. Learn MoreStarting at: $42.00
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PPDA
PPDA is a subtype-selective NMDA receptor antagonist that preferentially binds to NR2C/NR2D-containing receptors. Learn MoreStarting at: $119.00
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TC 1698 dihydrochloride
TC 1698 dihydrochloride is a selective nicotinic α7 receptor agonist that displays weak partial agonist/antagonist activity at β-subunit-containing receptors. Learn MoreStarting at: $125.00
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TCN 237 dihydrochloride
TCN 237 dihydrochloride is a highly potent NR2B-selective NMDA receptor antagonist that blocks NR2B-mediated calcium influx in Ltk cells with Ki value of 9.7 nM). Learn MoreStarting at: $115.00
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threo Ifenprodil hemitartrate
threo Ifenprodil hemitartrate is a potent σ receptor agonist and NR2B subunit-selective NMDA receptor antagonist. Learn MoreStarting at: $109.00
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DL-AP5
DL-AP5 is a potent NMDA antagonist. Learn MoreStarting at: $65.00
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N20C hydrochloride
N20C hydrochloride is a selective, non-competitive NMDA receptor antagonist that binds to the receptor-associated ion channel and prevents glutamate-induced Ca2+ influx. Learn MoreStarting at: $99.00
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MG 624
MG 624 inhibits α-Bgtx binding to chick α7 and α4β2 subtypes with Ki values of 106 nM and 84 μM respectively. Learn MoreStarting at: $99.00
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Synthalin sulfate
Synthalin sulfate is an effective non-competitive NMDA receptor antagonist in vivo and in vitro. Learn MoreStarting at: $85.00