Leukotriene and Related Receptors

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  • SR 2640 hydrochloride

    SR 2640 hydrochloride is a potent and selective competitive leukotriene D4 and E4 receptor antagonist,which Inhibits LTD4-, trachea contraction (pA2 = 8.7) and LTD4-attenuation of human PMN chemotaxis. Learn More

    Starting at: $95.00

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  • 5-Oxo-ETE

    5-Oxo-ETE is a potent oxoeicosanoid (OXE) receptor agonist (EC50 = 0.33 nM). Learn More

    Starting at: $179.00

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  • MK 571

    MK 571 is a potent CysLT1 (LTD4) leukotriene receptor inverse agonist (EC50 = 1.3 nM), which antagonizes LTD4-induced contractions of guinea pig trachea and ileum (pA2 values are 9.4 and 10.5 respectively). Learn More

    Starting at: $110.00

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  • Cinalukast

    Cinalukast is a potent, selective CysLT1 (LTD4) leukotriene receptor antagonist (IC50 = 6.4 nM), which inhibits LTD4-induced bronchoconstriction in guinea pigs when administered intravenously, orally or by aerosol. Learn More

    Starting at: $105.00

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  • BAY-u 9773

    BAY-u 9773 is a cysteinyl leukotriene receptor antagonist with equal affinity at both CysLT1 and CysLT2 receptors (pKB values are 6.8 and 6.5 respectively). Learn More

    Starting at: $95.00

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  • FPL 55712

    FPL 55712 is a leukotriene receptor antagonist which inhibits contraction of guinea pig trachealis induced by leukotrienes C4, D4, E4 and F4. Learn More

    Starting at: $149.00

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  • Leukotriene B4

    Leukotriene B4 is a potent lipid inflammatory mediator derived from the 5-lipoxygenase pathway of arachidonic acid metabolism. It binds to BLT1 and BLT2 receptors and acts as a potent chemotactic agent and activator of leukocytes. Learn More

    Starting at: $269.00

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  • LY 171883

    LY 171883 is a selective, orally active leukotriene D4 (LTD4) antagonist and also acts as an agonist at peroxisome proliferator-activated receptors (PPARs). Learn More

    Starting at: $75.00

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8 Item(s)

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