Esterases

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  • SGC-CBP30

    SGC-CBP30 is a potent CREBBP/EP300 bromodomain inhibitor (IC50 values are 21-69 and 38 nM for CREBBP and EP300 bromodomains respectively), which displays over 40-fold selectivity for CREBBP over BRD4(1). Learn More

    Starting at: $199.00

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  • VU 0155069

    VU 0155069 is a potent and selective phospholipase D1 (PLD1) inhibitor (IC50 values are 46 and 933 nM for PLD1 and PLD2 respectively), which inhibits migration of human and mouse breast cancer cell lines in transwell assays. Learn More

    Starting at: $130.00

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  • VU 0364739 hydrochloride

    VU 0364739 hydrochloride is a potent and selective phospholipase D2 (PLD2) inhibitor (IC50 = 20 nM) which displays 75-fold selectivity against PLD1 (IC50 = 1500 nM). Learn More

    Starting at: $155.00

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  • PACOCF3

    PACOCF3 is a phospholipase A2 inhibitor. Can also alter Ca2+ signaling in renal tubular cells. Learn More

    Starting at: $75.00

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  • U 73343

    U 73343 is an inactive analog of U 73122. Can be used as a negative control. Learn More

    Starting at: $85.00

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  • YM 26734

    YM 26734 is a competitive inhibitor of secretory phospholipase A2 (sPLA2) that exhibits a broad inhibitory profile to several sPLA2s (IC50 values are 0.2, 1, 1, 1 and 3 μM for sPLA2-X, -IIA, -IID, -V and -IIE respectively). Learn More

    Starting at: $135.00

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  • AACOCF3

    AACOCF3 is an inhibitor of cytosolic (85 kDa) phospholipase A2. It also inhibits fatty acid amide hydrolase (FAAH, anandamide amidase) in vitro. Learn More

    Starting at: $65.00

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  • m-3M3FBS

    m-3M3FBS is a activator of phospholipase C (PLC), which stimulates superoxide generation, Ca2+ release and inositol phosphate formation in a variety of cell types, and inhibits growth of the leukemic cell lines U937 and THP-1. Learn More

    Starting at: $98.00

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  • OBAA

    OBAA is a potent inhibitor of phospholipase A2 (IC50 = 70 nM), which reduces bronchospasm in guinea pigs in vivo. Learn More

    Starting at: $90.00

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  • o-3M3FBS

    o-3M3FBS is an inactive analog of m-3M3FBS. Used as a negative control. Learn More

    Starting at: $99.00

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  • LY 311727

    AM 630 is a CB2 antagonist/inverse agonist (Ki = 31.2 nM) that displays 165-fold selectivity over CB1 receptors. Learn More

    Starting at: $140.00

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  • Edelfosine

    Edelfosine is a synthetic lysophospholipid analog that selectively inhibits phosphatidylinositol phospholipase C. Learn More

    Starting at: $89.00

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  • STF 083010

    STF 083010 is an inhibitor of IRE1α endonuclease activity; blocks endogenous XBP1 mRNA splicing. Learn More

    Starting at: $119.00

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  • Physostigmine hemisulfate

    Physostigmine hemisulfate is a cholinesterase inhibitor. Learn More

    Starting at: $33.00

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  • Galanthamine hydrobromide

    Galanthamine hydrobromide is a long-acting, centrally active acetylcholinesterase inhibitor (IC50 = 410 nM) and allosteric potentiator at neuronal nicotinic ACh receptors. Learn More

    Starting at: $75.00

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  • Phenserine

    Phenserine is a Physostigmine analog that inhibits acetylcholinesterase.Phenserin also inhibits production of amyloid precursor protein (APP) and A&beta and improves morris water maze performance of scopolamine-treated rats. Learn More

    Starting at: $95.00

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  • PE 154

    PE 154 is a potent fluorescent inhibitor of human acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) (IC50 values are 280 pM and 16 nM respectively), which targets and labels β-amyloid plaques in histochemical analysis. Learn More

    Starting at: $160.00

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  • Rivastigmine tartrate

    Rivastigmine tartrate is a dual cholinesterase inhibitor (ChEI) which inhibits both butyrylcholinesterase (BChE) and acetylcholinesterase (AChE). Learn More

    Starting at: $70.00

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  • Acephate

    Anticholinesterase insecticide that produces cholinotoxicity, which displays weak inhibition of rat acetylcholinesterase (AChE) but potently inhibits cockroach AChE. Learn More

    Starting at: $59.00

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  • Tacrine hydrochloride

    AIDA is a relatively potent and selective antagonist of group I metabotropic glutamate receptors (mGlu1a), having no effect on group II (mGlu2) or group III (mGlu4) receptors expressed individually in baby hamster kidney cells. Learn More

    Starting at: $60.00

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