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SSR 69071
SSR 69071 is a high affinity, potent inhibitor of human leukocyte elastase (HLE) (IC50 = 3.9 nM), which displays species-selectivity (Ki values are 0.017, 1.70, 3.01, 58 and > 100 nM for human, mouse, rat, rabbit and porcine elastase respectively) and inhibits HLE-induced lung hemorrhage in mice (ID50 = 2.8 mg/kg) and reduces infarct size in an in vivo acute model of coronary ischemia-reperfusion injury. Orally active.
Additional Info
Additional Info
| Catalog No. | ES2682 |
|---|---|
| CAS Number | 344930-95-6 |
| Formula | C27H32N4O7S |
| M. Wt | 556.63 |
| Purity | >98 % |
| Solubility | Soluble to 10 mM in ethanol and to 25 mM in DMSO |
| Chemical Name | 2-[[6-Methoxy-4-(1-methylethyl)-1,1-dioxido-3-oxo-1,2-benzisothiazol-2(3H)-yl]methoxy]-9-[2-(1-piperidinyl)ethoxy]-4H-pyrido[1,2-a]pyrimidin-4-one |
| Synonyms | N/A |
| Storage | Store at +4°C |
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