D1 and D5 Receptors

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  • CY 208-243

    CY 208-243 is a centrally active dopamine D1 receptor agonist, selective over D2 receptor sites, which stimulates adenylate cyclase in rat striatal homogenates with an EC50 of 125 nM, that exerts antiParkinsonian activity in animal models. Learn More

    Starting at: $139.00

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  • SKF 83566 hydrobromide

    SKF 83566 hydrobromide is a potent and selective D1-like dopamine receptor antagonist (Ki~ 0.56 nM for D1; KB = 2 μM for D2). Learn More

    Starting at: $79.00

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  • SKF 38393 hydrobromide

    SKF 38393 hydrobromide is a prototypical D1-like dopamine receptor selective partial agonist. Learn More

    Starting at: $109.00

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  • SKF 83959 hydrobromide

    SKF 83959 hydrobromide is a dopamine D1-like receptor partial agonist that act as an antagonist in vivo, producing anti-Parkinsonian effects and antagonizing the behavioral effects of cocaine. Learn More

    Starting at: $139.00

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  • SKF 83822 hydrobromide

    SKF 83822 hydrobromide is a high affinity, selective dopamine D1-like receptor agonist. Learn More

    Starting at: $139.00

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  • SKF 81297 hydrobromide

    SKF 81297 hydrobromide is a dopamine D1-like receptor agonist. Learn More

    Starting at: $149.00

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  • Fenoldopam hydrochloride

    Fenoldopam hydrochloride is a selective D1-like dopamine receptor partial agonist with EC50 value of 57 nM. Learn More

    Starting at: $119.00

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  • LE 300

    LE 300 is a potent and selective dopamine D1 receptor antagonist (Ki values are 0.08 - 1.9 nM and 6 - 45 nM for D1 and D2 receptors respectively), which also displays moderate affinity for the 5-HT2A receptor (Ki = 20 nM). Active in vivo. Learn More

    Starting at: $139.00

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  • A 77636 hydrochloride

    A 77636 hydrochloride is a potent and selective dopamine D1-like receptor agonist (pEC50 values are 8.97 and < 5 for D1-like and D2-like receptors respectively), which displays anti-Parkinsonian activity following oral administration in vivo. Learn More

    Starting at: $140.00

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  • A 68930 hydrochloride

    A 68930 hydrochloride is a potent and selective D1-like dopamine receptor agonist (EC50 values are 2.1 and 3910 nM for D1-like and D2-like receptors respectively). Learn More

    Starting at: $115.00

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  • SCH 23390 hydrochloride

    SCH 23390 hydrochloride is a potent dopamine receptor antagonist (Ki values are 0.2 nM and 0.3 nM at D1 and D5 receptor sub-types respectively). Learn More

    Starting at: $90.00

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  • Dihydrexidine hydrochloride

    Dihydrexidine hydrochloride is a potent, full efficacy dopamine D1 agonist which shows no agonist activity at peripheral D2 receptors or adrenoceptors at doses which cause maximal stimulation of D1 sites. Learn More

    Starting at: $95.00

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  • SKF 77434 hydrobromide

    SKF 77434 hydrobromide is a selective dopamine D1-like receptor partial agonist (IC50 values are 19.7 and 2425 nM for binding to D1-like and D2-like receptors respectively). Learn More

    Starting at: $79.00

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  • LY 379268 disodium salt

    LY 379268 disodium salt is a sodium salt of LY 379268, a highly selective group II mGlu receptor agonist. Learn More

    Starting at: $295.00

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