AMPA Receptors

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  • CNQX disodium salt

    CNQX disodium salt is a more water soluble disodium salt of the AMPA/kainate antagonist CNQX . Learn More

    Starting at: $50.00

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  • 1-BCP

    1-BCP is a centrally active selective potentiator of AMPA-mediated responses. Learn More

    Starting at: $95.00

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  • Diazoxide

    Diazoxide is an antihypertensive, activates ATP-dependent K+ channels (Kir6), which induces activation of PKCε, an intermediate in the opening of mitoKATP channels, results in cardioprotection against hypoxia-induced death. Learn More

    Starting at: $55.00

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  • CMPDA

    CMPDA is a positive allosteric modulator of GluR2 receptors (EC50 values are 45.4 and 63.4 nM at GluR2i and GluR2o respectively, in a calcium influx screening assay), which binds at the modulator binding pocket located at the interdimer interface and the clamshell hinges. Learn More

    Starting at: $129.00

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  • (S)-CPW 399

    (S)-CPW 399 is a novel subtype-selective and weakly desensitizing AMPA receptor partial agonist (Ki values are 44, 109, 223, 1890 and 2090 nM at GluR5, GluR1, GluR2, GluR3 and GluR4 receptors respectively). Learn More

    Starting at: $139.00

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  • Philanthotoxin 74

    Philanthotoxin 74 is a subtype-selective AMPA receptor antagonist which inhibits homomeric GluR1, GluR3 and heteromeric GluR1/2 receptors. Learn More

    Starting at: $75.00

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  • ZK 200775

    Benzamil is a Na+/Ca2+ exhanger (NCX) inhibitor (IC50 ~ 100 nM); TRPP3 channel blocker (IC50 = 1.1 μM for inhibition of Ca2+-activated TRPP3 channel activity). Learn More

    Starting at: $140.00

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  • Talampanel

    L-371,257 is a potent, high affinity human oxytocin (OT) receptor antagonist (Ki = 4.6 nM) that displays > 800-fold selectivity over human arginine vasopressin receptors V1a and V2. Learn More

    Starting at: $125.00

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  • L-Quisqualic acid

    L-Quisqualic acid is a glutamate receptor agonist acting at AMPA receptors and metabotropic glutamate receptors positively linked to phosphoinositide hydrolysis. Learn More

    Starting at: $65.00

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  • UBP 282

    UBP 282 is an AMPA and kainate receptor antagonist. Learn More

    Starting at: $139.00

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  • (RS)-AMPA

    (RS)-AMPA is a prototypical and defining agonist for the AMPA subgroup of ionotropic glutamate receptors. Learn More

    Starting at: $139.00

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  • Piracetam

    Piracetam is a nootropic that displays cognitive enhancing properties.It facilitates efficiency of cholinergic neurotransmission at muscarinic receptors. Learn More

    Starting at: $55.00

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  • (RS)-AMPA hydrobromide

    (RS)-AMPA hydrobromide is a more water soluble hydrobromide salt of (RS)-AMPA. Learn More

    Starting at: $79.00

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  • (S)-AMPA

    (S)-AMPA is an active enantiomer of AMPA with an EC50 value of 3.5 μM. Learn More

    Starting at: $79.00

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  • (R)-AMPA

    (R)-AMPA is an inactive enantiomer of AMPA. Learn More

    Starting at: $229.00

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  • IEM 1925 dihydrobromide

    IEM 1925 dihydrobromide is a voltage- and use-dependent open-channel antagonist of AMPA receptors. Learn More

    Starting at: $109.00

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  • IDRA 21

    IDRA 21 is an inhibits AMPA receptor desensitization and enhances cognition by a related mechanism. Learn More

    Starting at: $119.00

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  • CX 546

    CX 546 is an AMPA receptor potentiator, which binds specifically to the agonist bound non-desensitized receptor, most likely destabilizing the desensitized receptor conformation. Learn More

    Starting at: $90.00

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  • CNQX

    CNQX is a potent AMPA/kainate receptor antagonist. Also antagonist at glycine modulatory site on NMDA receptor complex. Learn More

    Starting at: $95.00

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  • NBQX disodium salt

    NBQX disodium salt is a potent, selective and competitive AMPA receptor antagonist. Learn More

    Starting at: $75.00

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