Adenosine A1 Receptors

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  • DPCPX

    DPCPX is a potent and selective A1 adenosine receptor antagonist, both in vitro and in vivo. Learn More

    Starting at: $119.00

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  • PSB 36

    PSB 36 is a Potent and selective A1 adenosine receptor antagonist with binding affinities of 0.12, 187, 552, 6500 and 2300 nM for rA1, hA2B, rA2A, rA3 and hA3 receptors respectively. Learn More

    Starting at: $129.00

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  • N6-Cyclopentyladenosine

    N6-Cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist (Ki values are 2.3, 790 and 43 nM for human A1, A2A and A3 receptors respectively; EC50 = 18600 nM for hA2B). Learn More

    Starting at: $89.00

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  • 2-Chloro-N6-cyclopentyladenosine

    2-Chloro-N6-cyclopentyladenosine is a potent and selective adenosine A1 receptor agonist (Ki values are 0.8, 2300 and 42 nM for human A1, A2A and A3 receptors respectively; EC50 = 18800 nM for hA2B). Learn More

    Starting at: $99.00

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  • SLV 320

    SLV 320 is a potent and selective adenosine A1 receptor antagonist (Ki values are 1, 200, 398 and 3981 nM at human A1, A3, A2A and A2B receptors respectively). Learn More

    Starting at: $105.00

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  • 2'-MeCCPA

    2'-MeCCPA is a potent and highly selective agonist at A1 adenosine receptors (Ki values are 3.3, 9580, 37600 and 1150 nM for human recombinant A1, A2A, A2B and A3 receptors respectively), which acts as a full agonist and inhibits forskolin-stimulated adenylyl cyclase activity in rat cortical membranes with an IC50 value of 13.1 nM. Learn More

    Starting at: $189.00

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  • KW 3902

    KW 3902 is a selective adenosine A1 receptor antagonist; displays 890-fold selectivity for rat A1 receptors over A2A receptors (Ki values are 0.19 and 170 nM respectively). Learn More

    Starting at: $115.00

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  • PD 81723

    PD 81723 is an allosteric potentiator at the adenosine A1 receptor which acts via agonist-dependent and -independent mechanisms. Learn More

    Starting at: $95.00

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  • SDZ WAG 994

    SDZ WAG 994 is a potent and selective A1 adenosine receptor agonist (Ki values are 23, > 10000 and 25000 nM for A1, A2A and A2B receptors respectively). Learn More

    Starting at: $145.00

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  • GR 79236

    GR 79236 is a adenosine A1 receptor agonist (Ki = 3.1 nM). Learn More

    Starting at: $155.00

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  • (±)-5'-Chloro-5'-deoxy-ENBA

    (±)-5'-Chloro-5'-deoxy-ENBA is a highly selective adenosine A1 receptor agonist (Ki values are 0.51, 1290, 1340 and 2740 nM at A1, A3, A2A and A2B receptors respectively). Learn More

    Starting at: $135.00

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  • 1,3-Dipropyl-8-phenylxanthine

    1,3-Dipropyl-8-phenylxanthine is a selective A1 adenosine antagonist. Learn More

    Starting at: $95.00

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12 Item(s)

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