mAChR
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VU 0365114
VU 0365114 is a selective positive allosteric modulator of M5 (EC50 values are 2.7 μM for human M5, and >30 μM for M1, M2, M3 and M4 receptors). Learn MoreStarting at: $110.00
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VU 0238429
VU 0238429 is a selective positive allosteric modulator of M5 receptors (EC50 values are 1.16, >30 and >30 μM at M5, M1 and M3 receptors respectively), which displays no activity at M2 and M4 receptors. Learn MoreStarting at: $90.00
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Pilocarpine hydrochloride
Pilocarpine hydrochloride is a muscarinic agonist. Learn MoreStarting at: $49.00
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(+)-Muscarine iodide
(+)-Muscarine iodide is a muscarinic acetylcholine receptor agonist; mimics the activity of acetylcholine. Learn MoreStarting at: $155.00
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W-84 dibromide
W-84 dibromide stabilizes cholinergic antagonist-receptor complexes by an allosteric effect. Learn MoreStarting at: $98.00
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PTAC oxalate
PTAC oxalate is a muscarinic receptor ligand, which displays partial agonist activity at M2 and M4 receptors; exhibits antagonist effects at M1, M3 and M5 receptors (Ki values are 2.8, 0.2, 0.6, 0.2 and 0.8 nM respectively). Learn MoreStarting at: $139.00
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Oxotremorine sesquifumarate
Oxotremorine sesquifumarate is a muscarinic agonist. Learn MoreStarting at: $55.00
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Milameline hydrochloride
Muscarinic receptor agonist that displays roughly equal affinity at all receptor subtypes (Ki values are 2.3, 2.4, 3.6, 3.8 and 4.3 μM for hM1, hM2, hM3, hM4 and hM5 receptors respectively). Learn MoreStarting at: $95.00
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5-Methylfurmethiodide
5-Methylfurmethiodide is a potent muscarinic agonist. Learn MoreStarting at: $80.00
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Oxotremorine M
Oxotremorine M is a muscarinic receptor agonist. Learn MoreStarting at: $69.00