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7-TM Receptors
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AM 281
AM 281 is a potent, selective CB1 cannabinoid receptor antagonist/inverse agonist (Ki values are 12 and 4200 nM for CB1 and CB2 receptors respectively), which increases locomotor activity following systemic administration in vivo. Learn MoreStarting at: $140.00
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2'-MeCCPA
2'-MeCCPA is a potent and highly selective agonist at A1 adenosine receptors (Ki values are 3.3, 9580, 37600 and 1150 nM for human recombinant A1, A2A, A2B and A3 receptors respectively), which acts as a full agonist and inhibits forskolin-stimulated adenylyl cyclase activity in rat cortical membranes with an IC50 value of 13.1 nM. Learn MoreStarting at: $189.00
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AR-M 1000390 hydrochloride
AR-M 1000390 hydrochloride is a non-peptidic, low-internalizing δ-selective opioid receptor agonist; derivative of SNC 80. Learn MoreStarting at: $119.00
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ACEA
ACEA is a potent and highly selective CB1 receptor agonist (Ki = 1.4 nM) which displays >1400-fold selectivity over CB2 receptors. Learn MoreStarting at: $55.00
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LY 320135
LY 320135 is a potent CB1 receptor antagonist/inverse agonist (Ki = 141 nM) with greater than 70-fold selectivity over CB2 receptors (Ki > 10 μM). Learn MoreStarting at: $135.00
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(R)-(+)-Methanandamide
(R)-(+)-Methanandamide is a stable anandamide analog that is a selective agonist for the CB1 receptor (Ki values are 20 and 815 nM for CB1 and CB2 receptors respectively), which also displays agonist activity at vanilloid receptors. Learn MoreStarting at: $65.00
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SNC 80
SNC 80 is a highly selective and potent non-peptide δ-opioid agonist, 2000-fold selective over μ-opioid receptors. Learn MoreStarting at: $140.00
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TC-N 22A
TC-N 22A is a potent and selective mGlu4 receptor positive allosteric modulator (EC50 = 9 nM in human mGlu4-expressing BHK cells). Learn MoreStarting at: $135.00
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PD 81723
PD 81723 is an allosteric potentiator at the adenosine A1 receptor which acts via agonist-dependent and -independent mechanisms. Learn MoreStarting at: $95.00
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KW 3902
KW 3902 is a selective adenosine A1 receptor antagonist; displays 890-fold selectivity for rat A1 receptors over A2A receptors (Ki values are 0.19 and 170 nM respectively). Learn MoreStarting at: $115.00
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Alprenolol hydrochloride
Alprenolol hydrochloride is a β-adrenoceptor (β2 > β1 > β3) and 5-HT1A receptor antagonist. Learn MoreStarting at: $55.00
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Leelamine hydrochloride
Leelamine hydrochloride is a CB1 agonist which displaces binding of [3H]-SR141716A with an IC50 value of 2.86 μM. Learn MoreStarting at: $90.00
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A 77636 hydrochloride
A 77636 hydrochloride is a potent and selective dopamine D1-like receptor agonist (pEC50 values are 8.97 and < 5 for D1-like and D2-like receptors respectively), which displays anti-Parkinsonian activity following oral administration in vivo. Learn MoreStarting at: $140.00
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Telenzepine dihydrochloride
Telenzepine dihydrochloride is a selective high affinity muscarinic M1 receptor antagonist (Ki = 0.94 nM) which inhibits gastric acid secretion. Learn MoreStarting at: $50.00
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SB 205607 dihydrobromide
SB 205607 dihydrobromide is the first described non-peptide δ1 opioid receptor agonist with very high affinity and selectivity for the δ1 subtype (Ki values are 1.12, 2320 and 1790 nM at δ1, μ and κ receptors respectively). Learn MoreStarting at: $175.00
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DEA
DEA is a potent endocannabinoid and anandamide analog that activates CB1 receptors in microglia and binds to rat synaptosomal membranes (Ki = 34.4 nM). Learn MoreStarting at: $80.00
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BW 373U86
BW 373U86 is a potent, selective non-peptide δ-opioid receptor agonist. Learn MoreStarting at: $200.00
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NAS-181
NAS-181 is a potent, selective antagonist at the rat 5-HT1B receptor (Ki = 47 nM). Learn MoreStarting at: $155.00
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Org 12962 hydrochloride
Org 12962 hydrochloride is a selective 5-HT2C receptor agonist (pEC50 values are 7.01, 6.38 and 6.28 for 5-HT2C, 5-HT2A and 5-HT2B respectively), which displays antiaversive effects in a rat model of panic-like anxiety. Learn MoreStarting at: $105.00
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Antalarmin hydrochloride
Antalarmin hydrochloride is a non-peptide corticotropin-releasing hormone receptor 1 (CRF1) antagonist (Ki = 1 nM), which suppresses CRF-induced ACTH secretion and blocks CRF- and novelty-induced anxiety-like behavior in animal models of anxiety. Learn MoreStarting at: $140.00
